| 貨號 | 規格 | 價格 | 上海 | 北京 | 武漢 | 南京 | 購買數量 |
|---|---|---|---|---|---|---|---|
S84369-1mg |
99.6% | ￥600.00 | 10 | - | - | - |
|
S84369-5mg |
99.6% | ￥830.00 | 7 | - | - | - |
|
S84369-10mg |
99.6% | ￥1500.00 | 6 | - | - | - |
|
S84369-25mg |
99.6% | ￥2960.00 | 6 | - | - | - |
|
S84369-50mg |
≥98% | ￥5800.00 | 貨期：2-3天 | - | - | - |
|
S84369-100mg |
≥98% | ￥9800.00 | 貨期：2-3天 | - | - | - |
|
KDM4D-IN-1 is a new histone lysine demethylase 4D (KDM4D) inhibitor with an IC50 value of 0.41±0.03 μM
| 產品描述： | KDM4D-IN-1 is a new histone lysine demethylase 4D (KDM4D) inhibitor with an IC50 value of 0.41±0.03 μM | ||||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 靶點： | IC50:0.41±0.03 μM (KDM4D);HistoneDemethylase | ||||||||||||||||||||
| 體外研究： | KDM4D-IN-1 (Compound 10r) is the most potent one with an IC50 value of 0.41±0.03 μM against KDM4D. KDM4D-IN-1 displays almost no activity against KDM2B, KDM3B, and KDM5A (IC50>10 μM), indicating that KDM4D-IN-1 has a good selectivity for KDM4D against other selected KDMs | ||||||||||||||||||||
| 參考文獻： | 1. Fang Z, et al. Discovery of pyrazolo[1,5-a]pyrimidine-3-carbonitrile derivatives as a new class of histone lysine demethylase 4D (KDM4D) inhibitors. Bioorg Med Chem Lett. 2017 Jul 15;27(14):3201-3204. | ||||||||||||||||||||
| 溶解性： | Soluble in DMSO | ||||||||||||||||||||
| 保存條件： | -20℃ | ||||||||||||||||||||
| 配置溶液濃度參考： |
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| 注意： | 部分產品我司僅能提供部分信息，我司不保證所提供信息的權威性，僅供客戶參考交流研究之用。 |
上海工商
滬公網安備 31011702002021號
危險品化學品經營許可證（不帶存儲）
營業執照(三證合一)
北京