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KN-62是可滲透入細(xì)胞的CaM激酶II抑制劑,IC50為0.9 μM,直接與該酶的鈣調(diào)蛋白結(jié)合位點(diǎn)結(jié)合,同時(shí)還是非競(jìng)爭(zhēng)性P2X7受體拮抗劑,IC50為15 nM。A potent and selective inhibitor of CaMKII