產(chǎn)品描述: | TCS JNK 5a is a potent JNK3 inhibitor with a pIC50 of 6.7. TCS JNK 5a also inhibits JNK2 with a pIC50 of 6.5. |
靶點(diǎn): |
JNK3:6.7 (pIC50);JNK2:6.5 (pIC50) |
參考文獻(xiàn): |
1. Angell RM, et al. N-(3-Cyano-4,5,6,7-tetrahydro-1-benzothien-2-yl)amides as potent, selective, inhibitors of JNK2 and JNK3. Bioorg Med Chem Lett. 2007 Mar 1;17(5):1296-301. |
溶解性: |
DMSO : 20 mg/mL (60.16 mM; Need ultrasonic) |
保存條件: |
RT |
配置溶液濃度參考: |
|
1mg |
5mg |
10mg |
1 mM |
3.008 ml |
15.041 ml |
30.082 ml |
5 mM |
0.602 ml |
3.008 ml |
6.016 ml |
10 mM |
0.301 ml |
1.504 ml |
3.008 ml |
50 mM |
0.06 ml |
0.301 ml |
0.602 ml |
|
注意: |
部分產(chǎn)品我司僅能提供部分信息,我司不保證所提供信息的權(quán)威性,僅供客戶參考交流研究之用。 |